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1. A tribute to Prof. Stephen Hanessian (SH-1476YT)
Nicolas Moitessier and Vincent Mascitti
DOI: https://doi.org/10.24820/ark.5550190.p001.476
Full Text: PDF (360K)
pp. 1 - 3
published Jan 1 2019;
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2. Conformationally constrained fused bicyclic iminosugars: synthetic challenges and opportunities (SH-10872YR)
Raphaël Hensienne, Damien Hazelard and Philippe Compain
DOI: https://doi.org/10.24820/ark.5550190.p010.872
Full Text: PDF (2,389K)
pp. 4 - 43
received Jan 7 2019; accepted Feb 9 2019; published Feb 20 2019;
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3. Progress toward the total synthesis of mirabalin isomers (SH-10874VP)
Pierre-Georges Echeverria, Amandine Pons, Sébastien Prévost, Charlène Férard, Johan Cornil, Amandine Guérinot, Janine Cossy, Phannarath Phansavath and Virginie Ratovelomanana-Vidal
DOI: https://doi.org/10.24820/ark.5550190.p010.874
Full Text: PDF (1,888K)
pp. 44 - 68
received Jan 7 2019; accepted Feb 24 2019; published Feb 28 2019;
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4. 3-Alkylated indoles by reduction of sulfonyl indoles under flow chemical conditions (SH-10882YP)
Elena Chiurchiù, Alessandro Palmieri and Marino Petrini
DOI: https://doi.org/10.24820/ark.5550190.p010.882
Full Text: PDF (886K)
pp. 69 - 79
received Jan 18 2019; accepted Mar 7 2019; published Mar 12 2019;
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5. Synthetic studies toward eleganine A (SH-10897YP)
Christopher F. Cain, Evan H. Howard, Justin A. Goodwin and Juan R. Del Valle
DOI: https://doi.org/10.24820/ark.5550190.p010.897
Full Text: PDF (764K)
Supplementary Material: PDF (1,086K)
pp. 80 - 90
received Jan 30 2019; accepted Mar 7 2019; published Mar 13 2019;
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6. Ruthenium-catalyzed formation of pyrazoles or 3-hydroxynitriles from propargyl alcohols and hydrazines (SH-10893YP)
Julia Kaufmann, Elisabeth Jäckel and Edgar Haak
DOI: https://doi.org/10.24820/ark.5550190.p010.893
Full Text: PDF (668K)
Supplementary Material: PDF (1,551K)
pp. 91 - 101
received Jan 27 2019; accepted Mar 8 2019; published Mar 13 2019;
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7. Design of bis-NHC Ru-complexes featuring diarylmethylene N-substituents for olefin metathesis (SH-10894YP)
Idriss Curbet, Jennifer Morvan, Sophie Colombel-Rouen, Thierry Roisnel, Christophe Crévisy and Marc Mauduit
DOI: https://doi.org/10.24820/ark.5550190.p010.894
Full Text: PDF (1,321K)
Supplementary Material: PDF (3,702K)
pp. 102 - 112
received Jan 28 2019; accepted Mar 20 2019; published Apr 26 2019;
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8. Synthesis of nucleoside analogues using acyclic diastereoselective reactions (SH-10832YP)
Tommy Lussier, Marie-Ève Waltz, Garrett Freure, Philippe Mochirian, Starr Dostie, Michel Prévost and Yvan Guindon
DOI: https://doi.org/10.24820/ark.5550190.p010.832
Full Text: PDF (1,890K)
Supplementary Material: PDF (12,768K)
pp. 113 - 142
received Dec 3 2018; accepted Mar 11 2019; published Apr 29 2019;
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9. Comparison of affinity ranking by target-directed dynamic combinatorial chemistry and surface plasmon resonance (SH-10913YP)
Priska Frei, Marleen Silbermann, Tobias Mühlethaler, Xiaohua Jiang, Oliver Schwardt, Rachel Hevey and Beat Ernst
DOI: https://doi.org/10.24820/ark.5550190.p010.913
Full Text: PDF (1,772K)
Supplementary Material: PDF (3,172K)
pp. 143 - 167
received Feb 20 2019; accepted Apr 21 2019; published May 2 2019;
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10. A gram-scale synthesis of a macrocyclic amidinourea with strong antifungal activity through a Fukuyama tri-protected polyamine intermediate (SH-10895YP)
Matteo Borgini, Francesco Orofino, Giuseppina I. Truglio, Lorenzo Balestri and Maurizio Botta
DOI: https://doi.org/10.24820/ark.5550190.p010.895
Full Text: PDF (632K)
pp. 168 - 177
received Jan 30 2019; accepted May 4 2019; published May 16 2019;
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11. Fluorinated aminoglycosides (SH-10944YR)
Oscar M. Saavedra and Miguel A. Vilchis-Reyes
DOI: https://doi.org/10.24820/ark.5550190.p010.944
Full Text: PDF (1,994K)
pp. 178 - 226
received Apr 1 2019; accepted May 29 2019; published Jun 8 2019;
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12. Challenges of antibacterial drug discovery (SH-10955YR)
Folkert Reck, Johanna M. Jansen and Heinz E. Moser
DOI: https://doi.org/10.24820/ark.5550190.p010.955
Full Text: PDF (937K)
Supplementary Material: PDF (761K)
pp. 227 - 244
received Apr 11 2019; accepted Jun 17 2019; published Jul 12 2019;
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13. Synthesis of 2-substituted tetrahydroisoquinolin-6-ols: potential scaffolds for estrogen receptor modulation and/or microtubule degradation (SH-10962YP)
Tanya Mabank, Kabamba B. Alexandre, Stephen C. Pelly, Ivan R. Green and Willem A. L. van Otterlo
DOI: https://doi.org/10.24820/ark.5550190.p010.962
Full Text: PDF (1,159K)
pp. 245 - 279
received Apr 20 2019; accepted Jul 12 2019; published Jul 24 2019;
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14. Computational methods for prediction of drug properties - application to Cytochrome P450 metabolism prediction (SH-10970YR)
Mihai Burai Patrascu, Jessica Plescia, Amit Kalgutkar, Vincent Mascitti and Nicolas Moitessier
DOI: https://doi.org/10.24820/ark.5550190.p010.970
Full Text: PDF (993K)
pp. 280 - 298
received May 1 2019; accepted Jul 30 2019; published Oct 7 2019;
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