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1. Bio-transformation of FXR antagonist CDRI 80/574 (10-4951NP)
Alok K. Verma, Priti Khemaria, Jyoti Gupta, Dharmendra P. Singh, Bhawani S. Joshi, Raja Roy, Anjani K. Mishra and Ram Pratap
DOI: https://doi.org/10.3998/ark.5550190.0011.901
Full Text: PDF (1,067K)
Supplementary Material: PDF (8,232K)
pp. 1 - 11
received Jan 5 2010; accepted May 24 2010; published Jun 15 2010;
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2. Efficient preparation of novel N-propargylic β-enaminones from the reaction of β-alkoxyvinyltrihalomethyl[carboxy]ketones and propargylamines (10-4857GP)
Marcos A.P. Martins, Marcelo Rossatto, Liziê D. T. Prola, Dayse N. Moreira, Patrick T. Campos, Nilo Zanatta and Helio G. Bonacorso
DOI: https://doi.org/10.3998/ark.5550190.0011.902
Full Text: PDF (242K)
Supplementary Material: PDF (90K)
pp. 12 - 18
received Dec 11 2009; accepted Jun 2 2010; published Jun 16 2010;
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3. An efficient synthesis of functionalized 3-(hetaryl)pyrazoles (10-5190JP)
Ahmad S. Shawali, Thoraya A. Farghaly and Ahmad I. R. Aldahshoury
DOI: https://doi.org/10.3998/ark.5550190.0011.903
Full Text: PDF (443K)
pp. 19 - 30
received Mar 10 2010; accepted Jun 3 2010; published Jun 16 2010;
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4. Synthesis of conformationally constrained, orthogonally protected 3-azabicyclo[3.2.1]octane β-amino esters (10-5248VP)
Ferenc Fülöp, Brigitta Kazi, Lorand Kiss, Eniko Forro and Istvan Mandity
DOI: https://doi.org/10.3998/ark.5550190.0011.904
Full Text: PDF (457K)
pp. 31 - 39
received Mar 24 2010; accepted May 24 2010; published Jun 16 2010;
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5. The conformational diastereomers of 7-substituted-(8Z)-8-chloro-6,7-dihydro-9-(1,2-dihydro-6-R-naphthalen-4-yl)-2-R-5H-benzo[7]annulene, the question of atropisomerism versus ring inversion (10-4952QP)
Parviz Rashidi Ranjbar and Hamid Roshan
DOI: https://doi.org/10.3998/ark.5550190.0011.905
Full Text: PDF (584K)
pp. 40 - 53
received Jan 5 2010; accepted May 25 2010; published Jun 17 2010;
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6. Chiral lithium amide mediated asymmetric synthesis of 3-aryl-3,4-dihydroisocoumarins (10-4767MP)
Arvind Kumar Sharma, Yogita Maheshwary, Paramjit Singh and Kamal Nain Singh
DOI: https://doi.org/10.3998/ark.5550190.0011.906
Full Text: PDF (363K)
pp. 54 - 62
received Nov 21 2009; accepted Jun 3 2010; published Jun 18 2010;
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7. An inexpensive and efficient synthetic method for the preparation of pyromellitic dianhyride in ionic liquid (10-4307DP)
Lu Ming, Hu Yu Lin, Liu Xiao Bin, Zhang Sheng Bin, Ji Zhan Hui and Lu Ting Ting
DOI: https://doi.org/10.3998/ark.5550190.0011.907
Full Text: PDF (450K)
pp. 63 - 74
received Aug 10 2009; accepted Jun 7 2010; published Jun 18 2010;
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8. An efficient and versatile synthesis of 2, 2'-(alkanediyl)-bis-1H-benzimidazoles employing aqueous fluoroboric acid as catalyst: density functional theory calculations and fluorescence studies (10-5249QP)
Chhanda Mukhopadhyay, Sabari Ghosh and Ray J. Butcher
DOI: https://doi.org/10.3998/ark.5550190.0011.908
Full Text: PDF (651K)
Supplementary Material: PDF (2,478K)
pp. 75 - 96
received Mar 24 2010; accepted Jun 9 2010; published Jun 18 2010;
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9. Enhancing the helical distortion in pyrrolo[1,2-a]phenanthrolines (10-4953DP)
Florea Dumitrascu, Mino R. Caira, Constantin Draghici, Miron Teodor Caproiu, Loredana Barbu and Dan George Dumitrescu
DOI: https://doi.org/10.3998/ark.5550190.0011.909
Full Text: PDF (463K)
pp. 97 - 107
received Jan 5 2010; accepted May 28 2010; published Jun 18 2010;
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10. Orthogonally protected glycerols and 2-aminodiols, useful building blocks in heterocyclic chemistry (10-5304UP)
Isabelle Canet, Marie-Eve Sinibaldi, Anthony Ollivier, Marlène Goubert and Ahmatjan Tursun
DOI: https://doi.org/10.3998/ark.5550190.0011.910
Full Text: PDF (603K)
pp. 108 - 126
received Apr 15 2010; accepted May 31 2010; published Jun 19 2010;
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11. Condensed phase conformational isomerization of 5-[3-(1,3-dioxo-1,3-dihydro-isoindol-2-yl)-propoxy]-3-methyl-1H-pyrazole-4-carboxylic acid methyl ester (10-5075QP)
Ashish Kumar Tewari, Priyanka Srivastave, Ved Prakash Singh, Carmen Puerta and Pedro Valerga
DOI: https://doi.org/10.3998/ark.5550190.0011.911
Full Text: PDF (420K)
pp. 127 - 136
received Feb 6 2010; accepted May 31 2010; published Jun 20 2010;
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12. A simple and inexpensive procedure for low valent copper mediated benzylation of aldehydes in wet medium: synthesis of protease inhibitor synthon (10-4816QP)
Angshuman Chattopadhyay, Akhil Dubey and Dibakar Goswami
DOI: https://doi.org/10.3998/ark.5550190.0011.912
Full Text: PDF (210K)
pp. 137 - 145
received Dec 2 2009; accepted Jun 2 2010; published Jun 20 2010;
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13. A convenient synthesis of 1-(diethoxyphosphoryl)cyclopropanecarboxylates (10-5220CP)
Henryk Krawczyk, Katarzyna Wąsek, Jacek Kędzia, Jakub Wojciechowski and Wojciech M Wolf
DOI: https://doi.org/10.3998/ark.5550190.0011.913
Full Text: PDF (621K)
pp. 146 - 154
received Mar 17 2010; accepted Jun 2 2010; published Jun 20 2010;
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14. An efficient RuIII/BINAP catalytic system for the aldol reactions of ketones with various aldehydes (10-5156JP)
Khalil Tabatabaeian, Elahe Keshavarz, Manouchehr Mamaghani and Nosrat O. Mahmoodi
DOI: https://doi.org/10.3998/ark.5550190.0011.914
Full Text: PDF (273K)
pp. 155 - 162
received Mar 1 2010; accepted Jun 3 2010; published Jun 20 2010;
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15. A novel ionic liquid-supported Schiff base ligand applied in the Pd-catalyzed Suzuki–Miyaura coupling reaction (10-4886CP)
Yi-Qun Li, Bin Li and Jia Zheng
DOI: https://doi.org/10.3998/ark.5550190.0011.915
Full Text: PDF (349K)
pp. 163 - 170
received Dec 17 2009; accepted Jun 4 2010; published Jun 20 2010;
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16. Intramolecular cascade radical cyclizations promoted by samarium diiodide (10-5117OP)
Zhang Hu, Si-dong Li and Peng-zhi Hong
DOI: https://doi.org/10.3998/ark.5550190.0011.916
Full Text: PDF (406K)
pp. 171 - 177
received Feb 19 2010; accepted Jun 20 2010; published Jul 3 2010;
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17. An efficient oxidation of 2-pyrazolines and isoxazolines by bis-bromine-1,4-diazabicyclo[2.2.2]octane complex (DABCO-Br2) (10-4311MP)
Davood Azarifar, Kaveh Khosravi and Rahman Ali Veisi
DOI: https://doi.org/10.3998/ark.5550190.0011.917
Full Text: PDF (563K)
pp. 178 - 184
received Aug 12 2009; accepted Jun 20 2010; published Jul 3 2010;
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18. Amino acid derivatives. Part 5. Synthesis and anti-HIV activity of new sebacoyl precursor derived thioureido-amino acid and phthalimide derivatives (10-5081MP)
Najim A. Al-Masoudi, Nahed Al-Haidery, Naeem T. Faili and C. Pannecouque
DOI: https://doi.org/10.3998/ark.5550190.0011.918
Full Text: PDF (474K)
pp. 185 - 195
received Feb 7 2010; accepted Jun 18 2010; published Jul 7 2010;
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19. Synthesis and antimicrobial activities of novel peptide deformylase inhibitors (10-3973MP)
Ling Yin, Wei-Ren Xu, Zhi-Guo Wang, Da-Tong Zhang, Jiong Jia, Yan-Qing Ge, Yan Li and Jian-Wu Wang
DOI: https://doi.org/10.3998/ark.5550190.0011.919
Full Text: PDF (553K)
Supplementary Material: PDF (496K)
pp. 196 - 205
received Apr 7 2009; accepted Jun 18 2010; published Jul 7 2010;
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20. A practical synthesis of a novel PPAR alpha agonist (10-5349KP)
Joel Slade, Hui Liu, Mahavir Prashad and Kapa Prasad
DOI: https://doi.org/10.3998/ark.5550190.0011.920
Full Text: PDF (461K)
pp. 206 - 215
received Apr 28 2010; accepted Jun 17 2010; published Jul 7 2010;
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21. Convenient and robust one-pot synthesis of symmetrical and unsymmetrical benzyl thioethers from benzyl halides using thiourea (10-4802SP)
Kevin S. Eccles, Curtis J. Elcoate, Simon E. Lawrence and Anita R. Maguire
DOI: https://doi.org/10.3998/ark.5550190.0011.921
Full Text: PDF (410K)
pp. 216 - 228
received Nov 30 2009; accepted Jun 16 2010; published Jul 7 2010;
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22. Organocatalytic asymmetric conjugate addition of cyclic 1,3-dicarbonyl compounds to β,γ-unsaturated α-ketoesters (10-5234UP)
Jin-jia Wang, Jin-hua Lao, Zhi-peng Hu, Rui-Jiong Lu, Shao-zhen Nie, Quan-sheng Du and Ming Yan
DOI: https://doi.org/10.3998/ark.5550190.0011.922
Full Text: PDF (747K)
pp. 229 - 243
received Mar 20 2010; accepted Jun 20 2010; published Jul 7 2010;
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23. The synthesis of new thiosubstituted butadienes, butenynes and butatrienes (10-4752CP)
Cemil Ibis and Neslihan Beyazit
DOI: https://doi.org/10.3998/ark.5550190.0011.923
Full Text: PDF (718K)
pp. 244 - 256
received Nov 18 2009; accepted May 28 2010; published Jul 9 2010;
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24. Experimental and DFT study of 2-ferrocenylpropan-2-ol cyclodimerization products (10-5222HP)
Jasmina Lapić, Mario Cetina, Davor Šakić, Senka Djaković, Valerije Vrček and Vladimir Rapić
DOI: https://doi.org/10.3998/ark.5550190.0011.924
Full Text: PDF (1,065K)
Supplementary Material: PDF (188K)
pp. 257 - 268
received Mar 17 2010; accepted May 31 2010; published Jul 9 2010;
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25. A study of [1]benzofuro[3,2-c]pyridine derivatives (10-5279UP)
Denisa Tarabová, Ján Titiš, Naďa Prónayová, Anton Gatial and Alžbeta Krutošíková
DOI: https://doi.org/10.3998/ark.5550190.0011.925
Full Text: PDF (1,039K)
pp. 269 - 281
received Apr 6 2010; accepted Jun 2 2010; published Jul 9 2010;
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26. A facial synthesis of quinazolino[1,4]benzodiazepine alkaloids via reductive N-heterocyclization of N-(2-nitrobenzoyl)amides: total synthesis of asperlicin C, circumdatin H, and its analogues (10-4137MP)
Naim H. Al-Said, Khaled Q. Shawakfeh, Mohammad I. Ibrahim and Sami H. Tayyem
DOI: https://doi.org/10.3998/ark.5550190.0011.926
Full Text: PDF (245K)
pp. 282 - 292
received Jun 6 2009; accepted Jun 20 2010; published Jul 11 2010;
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27. Selective alkylation of aminophenols (10-5213GP)
Jiaxi Xu and Renchao Wang
DOI: https://doi.org/10.3998/ark.5550190.0011.927
Full Text: PDF (210K)
pp. 293 - 299
received Mar 15 2010; accepted Jul 2 2010; published Jul 19 2010;
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28. Microwave-assisted one-pot reactions for direct synthesis of 6-methylpurines (10-4832OP)
Hai-Ming Guo, Zhi-Jie Mao, Hong-Ying Niu, Dong-Chao Wang, Gui-Sheng Zhang and Gui-Rong Qu
DOI: https://doi.org/10.3998/ark.5550190.0011.928
Full Text: PDF (348K)
pp. 300 - 307
received Dec 5 2009; accepted Jun 22 2010; published Jul 19 2010;
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29. Nucleophilic substitution reactions, molecular aggregation, structure and lipophilicity of 6-chloro-3-chloromethyl-1,2,4-triazolo[4,3-b]pyridazine (10-5347HP)
Anna Katrusiak and Andrzej Katrusiak
DOI: https://doi.org/10.3998/ark.5550190.0011.929
Full Text: PDF (684K)
pp. 308 - 318
received Apr 27 2010; accepted Jun 23 2010; published Jul 19 2010;
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30. Microwave-assisted C-C cross-coupling reactions of aryl and heteroaryl halides in water (10-5361DP)
Kamal M. Dawood and Moteaa M. El-Deftar
DOI: https://doi.org/10.3998/ark.5550190.0011.930
Full Text: PDF (334K)
pp. 319 - 330
received May 1 2010; accepted Jul 21 2010; published Jul 27 2010;
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